Search Result "inverse agonists"


Histamine H3-Receptor Inverse Agonists as Novel Antipsychotics

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2009 Page: 132-136
Author(s): Chihiro Ito

Review Article

Advances in Medicinal Chemistry of Estrogen-related Receptor Alpha (ERRα) Inverse Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 23 Issue: 20 Year: 2023 Page: 1952-1963
Author(s):

Novel Benzimidazole Derivatives as Selective CB2 Inverse Agonists

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 5 Year: 2006 Page: 298-303
Author(s): D. Page, M.-C. Brochu, H. Yang, W. Brown, S. St-Onge, E. Martin, D. Salois

Review Article

Advances in the Understanding of the Cannabinoid Receptor 1 – Focusing on the Inverse Agonists Interactions

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 1 Year: 2019 Page: 1908-1919
Author(s): Silvana Russo,Walter Filgueira De Azevedo

Review Article

δ Opioid Receptor Inverse Agonists and their In Vivo Pharmacological Effects

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 3 Year: 2020 Page: 2889-2902
Author(s): Shigeto Hirayama,Hideaki Fujii

Angiotensin II Receptor Blocker as an Inverse Agonist: A Current Perspective

Journal: Current Hypertension Reviews
Volume: 1 Issue: 2 Year: 2005 Page: 115-121
Author(s): Shin-ichiro Miura, Masahiro Fujino, Keijiro Saku

Histamine H3 Receptor (H3R) Antagonists and Inverse Agonists in the Treatment of Sleep Disorders

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 1 Year: 2011 Page: 1426-1429
Author(s): Meredith Broderick, Tony Masri

5-HT2A Inverse-Agonists for the Treatment of Insomnia

Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 969-976
Author(s): Bradley R. Teegarden, Hussien Al Shamma, Yifeng Xiong

The Evolution of Histamine H3 Antagonists/Inverse Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 648-660
Author(s): Evan P. Lebois, Carrie K. Jones, Craig W. Lindsley

Assessing Receptor Affinity for Inverse Agonists: Schild and Cheng-Prusoff Methods Revisited

Journal: Current Drug Targets
Volume: 8 Issue: 1 Year: 2007 Page: 197-202
Author(s): Jesus Giraldo, Juan Serra, David Roche, Xavier Rovira

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